|
|
|
5-HT1A receptor
|
|
|
Hs |
Agonist |
Full agonist |
9.4 – 10.3 |
pKi |
- |
22-25 |
|
⤷ |
pKi
9.4 – 10.3
[22-25]
|
5-HT7 receptor
|
|
|
Rn |
Agonist |
Full agonist |
9.5 – 9.9 |
pKi |
- |
29-30 |
|
⤷ |
pKi
9.5 – 9.9
[29-30]
|
5-HT7 receptor
|
|
|
Hs |
Agonist |
Full agonist |
9.0 – 10.0 |
pKi |
- |
4,11,14,31 |
|
⤷ |
pKi
9.0 – 10.0
[4,11,14,31]
|
5-HT7 receptor
|
|
|
Mm |
Agonist |
Full agonist |
9.0 |
pKi |
- |
27 |
|
⤷ |
pKi
9.0
[27]
|
5-HT1D receptor
|
|
|
Hs |
Agonist |
Full agonist |
8.6 – 9.2 |
pKi |
- |
10,16,33 |
|
⤷ |
pKi
8.6 – 9.2
[10,16,33]
|
5-HT1B receptor
|
|
|
Hs |
Agonist |
Full agonist |
7.7 – 8.8 |
pKi |
- |
26,33 |
|
⤷ |
pKi
7.7 – 8.8
[26,33]
|
5-HT1B receptor
|
|
|
Mm |
Agonist |
Full agonist |
8.1 |
pKi |
- |
18 |
|
⤷ |
pKi
8.1
[18]
|
5-HT5A receptor
|
|
|
Rn |
Agonist |
Full agonist |
7.9 |
pKi |
- |
8 |
|
⤷ |
pKi
7.9
[8]
|
5-HT5A receptor
|
|
|
Hs |
Agonist |
Full agonist |
7.6 – 7.7 |
pKi |
- |
9,28 |
|
⤷ |
pKi
7.6 – 7.7
[9,28]
|
5-HT5A receptor
|
|
|
Mm |
Agonist |
Full agonist |
7.3 – 7.8 |
pKi |
- |
9,19,34 |
|
⤷ |
pKi
7.3 – 7.8
[9,19,34]
|
5-HT2B receptor
|
|
|
Hs |
Agonist |
Full agonist |
6.7 – 6.9 |
pKi |
- |
12,15 |
|
⤷ |
pKi
6.7 – 6.9
[12,15]
|
5-HT2B receptor
|
|
|
Rn |
Agonist |
Full agonist |
6.8 |
pKi |
- |
15,32 |
|
⤷ |
pKi
6.8
[15,32]
|
5-HT2A receptor
|
|
|
Hs |
Agonist |
Full agonist |
6.5 |
pKi |
- |
12 |
|
⤷ |
pKi
6.5
[12]
|
5-HT1F receptor
|
|
|
Hs |
Agonist |
Full agonist |
6.1 |
pKi |
- |
1-2 |
|
⤷ |
pKi
6.1
[1-2]
|
5-HT6 receptor
|
|
|
Hs |
Agonist |
Full agonist |
6.1 |
pKi |
- |
13 |
|
⤷ |
pKi
6.1
[13]
|
5-HT6 receptor
|
|
|
Rn |
Agonist |
Full agonist |
5.5 – 6.7 |
pKi |
- |
5-6,21 |
|
⤷ |
pKi
5.5 – 6.7
[5-6,21]
|
5-HT2C receptor
|
|
|
Hs |
Agonist |
Full agonist |
5.2 – 6.7 |
pKi |
- |
7,12 |
|
⤷ |
pKi
5.2 – 6.7
[7,12]
|
5-ht1e receptor
|
|
|
Hs |
Agonist |
Full agonist |
5.1 – 5.5 |
pKi |
- |
2-3,20,26 |
|
⤷ |
pKi
5.1 – 5.5
[2-3,20,26]
|
5-HT1F receptor
|
|
|
Rn |
Agonist |
Full agonist |
5.6 |
pIC50 |
- |
17 |
|
⤷ |
pIC50
5.6
[17]
|
|