Synonyms: compound 39 [PMID: 36367749]
Compound class:
Synthetic organic
Comment: MRS8054 is a positive allosteric modulator of the adenosine A3 receptor [1]. It is orally bioavailable in rat.
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Bioactivity Comments |
MRS8054 enhances Cl-IB-MECA-stimulated [35S]GTPγS binding in vitro [1]. |
Selectivity at GPCRs | ||||||||||||||||||||||||||||||||||
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