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CCK-58   Click here for help

GtoPdb Ligand ID: 3552

Compound class: Endogenous peptide in human, mouse or rat
Species: Human
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Natural/Endogenous Targets
Target
CCK1 receptor
Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference
CCK1 receptor Ligand is endogenous in the given species Hs Agonist Agonist - - -
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Additional information and targets (data relate to human unless otherwise stated)
Description Data Reference
Potency order of endogenous ligands at CCK2 receptor CCK-8 (CCK, P06307), CCK-39 (CCK, P06307), CCK-33 (CCK, P06307), CCK-58 (CCK, P06307) ≥ gastrin-17 (GAST, P01350), desulfated cholecystokinin-8, CCK-4 (CCK, P06307)
Potency order of endogenous ligands at CCK1 receptor CCK-8 (CCK, P06307), CCK-58 (CCK, P06307), CCK-39 (CCK, P06307), CCK-33 (CCK, P06307) >> gastrin-17 (GAST, P01350), desulfated cholecystokinin-8 > CCK-4 (CCK, P06307)
Ligand mentioned in the following text fields
Cholecystokinin receptors overview