View and download lists of GPCR targets:

View a list of class A GPCRs, class B GPCRs, class C GPCRs, class frizzled GPCRs, adhesion class GPCRs or other 7TM proteins

Families that contain targets of relevance to immunopharmacology are highlighted in blue

• G protein-coupled receptors C
  • Orphan and other 7TM receptors
  • 5-Hydroxytryptamine receptors C
  • Acetylcholine receptors (muscarinic) C
  • Adenosine receptors C
  • Adhesion Class GPCRs C
  • Adrenoceptors C
  • Angiotensin receptors C
  • Apelin receptor C
  • Bile acid receptor C
  • Bombesin receptors C
  • Bradykinin receptors C
  • Calcitonin receptors C
  • Calcium-sensing receptor C
  • Cannabinoid receptors C
  • Chemerin receptors C
  • Chemokine receptors C
  • Cholecystokinin receptors C
  • Class A Orphans C
    • Class A Orphans with no pharmacology C
    • Class A Orphans with only surrogate ligands C
    • Class A Orphans with emerging pharmacology C
    • GPR18, GPR55 and GPR119 C
    • GPR42, GPR84 C
    • LGR4, LGR5, LGR6 C
    • Mas1, BB3/brs3, GPR17 C
    • TAAR2, TAAR3, TAAR4p, TAAR5, TAAR6, TAAR8, TAAR9 C
  • Class B Orphans
  • Class C Orphans C
  • Class Frizzled GPCRs C
  • Complement peptide receptors C
  • Corticotropin-releasing factor receptors C
  • Dopamine receptors C
  • Endothelin receptors C
  • Formylpeptide receptors C
  • Free fatty acid receptors C
  • G protein-coupled estrogen receptor C
  • GABA_B receptors C
  • Galanin receptors C
  • Ghrelin receptor C
  • Glucagon receptor family C
  • Glycoprotein hormone receptors C
  • Gonadotrophin-releasing hormone receptors C
  • GPR143 C
  • GPR18, GPR55 and GPR119 C
  • Histamine receptors C
  • Hydroxycarboxylic acid receptors C
  • Kisspeptin receptor C
  • Leukotriene receptors C
  • Lysophospholipid (LPA) receptors C
  • Lysophospholipid (S1P) receptors C
  • Melanin-concentrating hormone receptors C
  • Melanocortin receptors C
  • Melatonin receptors C
  • Metabotropic glutamate receptors C
  • Motilin receptor C
  • Neuromedin U receptors C
  • Neuropeptide FF/neuropeptide AF receptors C
  • Neuropeptide S receptor C
  • Neuropeptide W/neuropeptide B receptors C
  • Neuropeptide Y receptors C
  • Neurotensin receptors C
  • Opioid receptors C
  • Opsin receptors C
  • Orexin receptors C
  • Oxoglutarate receptor C
  • P2Y receptors C
  • Parathyroid hormone receptors C
  • Platelet-activating factor receptor C
  • Prokineticin receptors C
  • Prolactin-releasing peptide receptor C
  • Prostanoid receptors C
  • Proteinase-activated receptors C
  • QRFP receptor C
  • Relaxin family peptide receptors C
  • Somatostatin receptors C
  • Succinate receptor C
  • Tachykinin receptors C
  • Taste 1 receptors C
  • Taste 2 receptors C
  • Thyrotropin-releasing hormone receptors C
  • Trace amine receptor C
  • Urotensin receptor C
  • Vasopressin and oxytocin receptors C
  • VIP and PACAP receptors C
  • Other non-GPCR 7TM proteins C