tesevatinib [Ligand Id: 7944] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| epidermal growth factor receptor in Human [GtoPdb: 1797] [UniProtKB: P00533] | ||||||||
| GtoPdb | - | - | 9.52 | pIC50 | 0.3 | nM | IC50 | Clin Cancer Res (2007) 13: 3713-23 [PMID:17575237] |
| kinase insert domain receptor in Human [GtoPdb: 1813] [UniProtKB: P35968] | ||||||||
| GtoPdb | - | - | 8.82 | pIC50 | 1.5 | nM | IC50 | Clin Cancer Res (2007) 13: 3713-23 [PMID:17575237] |
| fms related receptor tyrosine kinase 4 in Human [GtoPdb: 1814] [UniProtKB: P35916] | ||||||||
| GtoPdb | - | - | 8.06 | pIC50 | 8.7 | nM | IC50 | Clin Cancer Res (2007) 13: 3713-23 [PMID:17575237] |
| EPH receptor B4 in Human [GtoPdb: 1833] [UniProtKB: P54760] | ||||||||
| GtoPdb | - | - | 8.85 | pIC50 | 1.4 | nM | IC50 | Clin Cancer Res (2007) 13: 3713-23 [PMID:17575237] |
| erb-b2 receptor tyrosine kinase 2 in Human [GtoPdb: 2019] [UniProtKB: P04626] | ||||||||
| GtoPdb | - | - | 7.8 | pIC50 | 16 | nM | IC50 | Clin Cancer Res (2007) 13: 3713-23 [PMID:17575237] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
