XRD-0394 [Ligand Id: 13457] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| ATM serine/threonine kinase in Human [GtoPdb: 1934] [UniProtKB: Q13315] | ||||||||
| GtoPdb | - | - | 8.61 | pIC50 | 2.43 | nM | IC50 | WO2021022078A1. Dual atm and dna-pk inhibitors for use in anti-tumor therapy (2021) |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha in Human [GtoPdb: 2153] [UniProtKB: P42336] | ||||||||
| GtoPdb | - | - | 7.8 | pIC50 | 16 | nM | IC50 | WO2021022078A1. Dual atm and dna-pk inhibitors for use in anti-tumor therapy (2021) |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta in Human [GtoPdb: 2155] [UniProtKB: O00329] | ||||||||
| GtoPdb | - | - | 7.14 | pIC50 | 73 | nM | IC50 | WO2021022078A1. Dual atm and dna-pk inhibitors for use in anti-tumor therapy (2021) |
| protein kinase, DNA-activated, catalytic subunit in Human [GtoPdb: 2800] [UniProtKB: P78527] | ||||||||
| GtoPdb | - | - | 9.2 | pIC50 | 0.63 | nM | IC50 | WO2021022078A1. Dual atm and dna-pk inhibitors for use in anti-tumor therapy (2021) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
