compound 4d [PMID: 38746883] [Ligand Id: 13365] activity data from GtoPdb

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  • cathepsin L in Human [GtoPdb: 2351] [UniProtKB: P07711]
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  • cathepsin S in Human [GtoPdb: 2353] [UniProtKB: P25774]
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  • CoV 3C-like (main) protease in SARS-CoV-2 [GtoPdb: 3111]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
cathepsin L in Human [GtoPdb: 2351] [UniProtKB: P07711]
GtoPdb - - 6.15 pIC50 701 nM IC50 ACS Med Chem Lett (2024) 15: 602-609 [PMID:38746883]
cathepsin S in Human [GtoPdb: 2353] [UniProtKB: P25774]
GtoPdb - - 9.15 pIC50 0.7 nM IC50 ACS Med Chem Lett (2024) 15: 602-609 [PMID:38746883]
CoV 3C-like (main) protease in SARS-CoV-2 [GtoPdb: 3111]
GtoPdb - - 5.26 pIC50 5540 nM IC50 ACS Med Chem Lett (2024) 15: 602-609 [PMID:38746883]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.