Compound class:
Synthetic organic
Comment: Positive allosteric modulator of the human A3 adenosine receptor.
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References |
1. Heitman LH, Göblyös A, Zweemer AM, Bakker R, Mulder-Krieger T, van Veldhoven JP, de Vries H, Brussee J, Ijzerman AP. (2009)
A series of 2,4-disubstituted quinolines as a new class of allosteric enhancers of the adenosine A3 receptor. J Med Chem, 52 (4): 926-31. [PMID:19161279] |