Compound class:
Synthetic organic
Comment: Compound A is a selective agonist of the free fatty acid receptor 4 (FFA4R) [1]. The compound is a small molecule, orally active mimic of ω-3-fatty acids, the endogenous ligands of FFA4R [2].
![]() Ligand Activity Visualisation ChartsThese are box plot that provide a unique visualisation, summarising all the activity data for a ligand taken from ChEMBL and GtoPdb across multiple targets and species. Click on a plot to see the median, interquartile range, low and high data points. A value of zero indicates that no data are available. A separate chart is created for each target, and where possible the algorithm tries to merge ChEMBL and GtoPdb targets by matching them on name and UniProt accession, for each available species. However, please note that inconsistency in naming of targets may lead to data for the same target being reported across multiple charts. ✖ |
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Bioactivity Comments |
CpdA acts as a potent anti-inflammatory agent in vitro and in vivo, and improves glucose tolerance (and other diabetes related parameters) in a mouse model of type 2 diabetes [1]. |
Selectivity at GPCRs | ||||||||||||||||||||||||||||||||||
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