PMX205   Click here for help

GtoPdb Ligand ID: 5762

Synonyms: PMX 205 | PMX-205
Immunopharmacology Ligand
Comment: PMX205 is potent, non-competitive and orally active C5a receptor peptide antagonist [4].
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
C5a1 receptor Hs Antagonist Antagonist 7.5 pIC50 - 2-3
pIC50 7.5 (IC50 3.1x10-8 M) [2-3]