chemerin   Click here for help

GtoPdb Ligand ID: 2945

Synonyms: RARRES2 | retinoic acid receptor responder protein 2 | TIG2
Species: Human
Click here for help
Natural/Endogenous Targets
Target
chemerin receptor 1
chemerin receptor 2
Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference
chemerin receptor 1 Ligand is endogenous in the given species Hs Agonist Full agonist 8.3 pKd - 1
pKd 8.3 (Kd 4.9x10-9 M) [1]
chemerin receptor 2 Ligand is endogenous in the given species Hs Agonist Full agonist 8.3 pKd - 1
pKd 8.3 (Kd 5.3x10-9 M) [1]
chemerin receptor 2 Ligand is endogenous in the given species Hs Agonist Full agonist 8.8 – 9.6 pEC50 - 1,3
pEC50 8.8 – 9.6 (EC50 2.4x10-10 M) [1,3]
chemerin receptor 1 Ligand is endogenous in the given species Hs Agonist Full agonist 7.6 – 8.5 pEC50 - 1-5
pEC50 7.6 – 8.5 (EC50 4.5x10-9 – 3x10-9 M) [1,3-5]
pEC50 8.0 (EC50 9.7x10-9 M) [2]
Description: In a β-arrestin recruitment assay.
Ligand mentioned in the following text fields