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ChEMBL ligand: CHEMBL464108 |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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phosphodiesterase 4A in Human [GtoPdb: 1300] [UniProtKB: P27815] | ||||||||
GtoPdb | Inhibition of PDE4A1A activity in vitro. | - | 5.12 | pIC50 | 7510 | nM | IC50 | Free Radic. Biol. Med. (2017) 106: 379-392 [PMID:28263828] |
phosphodiesterase 4B in Human [GtoPdb: 1301] [UniProtKB: Q07343] | ||||||||
GtoPdb | Inhibition of PDE4B2 activity in vitro. | - | 5.07 | pIC50 | 8580 | nM | IC50 | Free Radic. Biol. Med. (2017) 106: 379-392 [PMID:28263828] |
phosphodiesterase 4C in Human [GtoPdb: 1302] [UniProtKB: Q08493] | ||||||||
GtoPdb | Inhibition of PDE4C1 activity in vitro. | - | 5.76 | pIC50 | 1750 | nM | IC50 | Free Radic. Biol. Med. (2017) 106: 379-392 [PMID:28263828] |
phosphodiesterase 4D in Human [GtoPdb: 1303] [UniProtKB: Q08499] | ||||||||
GtoPdb | Inhibition of PDE4D2 activity in vitro. | - | 5.45 | pIC50 | 3530 | nM | IC50 | Free Radic. Biol. Med. (2017) 106: 379-392 [PMID:28263828] |
ChEMBL data shown on this page come from version 27:
Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]