petesicatib [Ligand Id: 9855] activity data from GtoPdb

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  • cathepsin V in Human [GtoPdb: 2352] [UniProtKB: O60911]
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  • cathepsin S in Human [GtoPdb: 2353] [UniProtKB: P25774]
  • cathepsin S in Mouse [GtoPdb: 2353] [UniProtKB: O70370]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
cathepsin V in Human [GtoPdb: 2352] [UniProtKB: O60911]
GtoPdb - - 6.15 pIC50 700 nM IC50 Sci Rep (2017) 7: 2775 [PMID:28584258]
cathepsin S in Human [GtoPdb: 2353] [UniProtKB: P25774]
GtoPdb - - 10 pIC50 0.1 nM IC50 Sci Rep (2017) 7: 2775 [PMID:28584258]
cathepsin S in Mouse [GtoPdb: 2353] [UniProtKB: O70370]
GtoPdb - - 9.52 pIC50 0.3 nM IC50 Sci Rep (2017) 7: 2775 [PMID:28584258]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.