Galapagos MAPKAPK5 inhibitor D [Ligand Id: 9848] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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| MAPK activated protein kinase 5 in Human [GtoPdb: 2096] [UniProtKB: Q8IW41] | ||||||||
| GtoPdb | - | - | 7.43 | pIC50 | 37 | nM | IC50 | Discovery of inhibitors of MAPKAPK5, a novel target for rheumatoid arthritis. www.rsc.org |
| GtoPdb | Binned IC50 range from patent. | - | 9 | pIC50 | 1 | nM | IC50 | WO2007138072A2. Triazolopyrazine compounds useful for the treatment of degenerative & inflammatory diseases (2007) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
