STK16-IN-1 [Ligand Id: 9692] activity data from GtoPdb

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  • mechanistic target of rapamycin kinase in Human [GtoPdb: 2109] [UniProtKB: P42345]
Created with Highcharts 10.3.3ValuesChart context menumechanistic target of rapamycin kinasepKd HumanpKi HumanpIC50 HumanpEC50 Human0123456Highcharts.com
  • phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta in Human [GtoPdb: 2155] [UniProtKB: O00329]
Created with Highcharts 10.3.3ValuesChart context menuphosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit deltapKd HumanpKi HumanpIC50 HumanpEC50 Human01234567Highcharts.com
  • phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma in Human [GtoPdb: 2156] [UniProtKB: P48736]
Created with Highcharts 10.3.3ValuesChart context menuphosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gammapKd HumanpKi HumanpIC50 HumanpEC50 Human01234567Highcharts.com
  • serine/threonine kinase 16 in Human [GtoPdb: 2213] [UniProtKB: O75716]
Created with Highcharts 10.3.3ValuesChart context menuserine/threonine kinase 16pKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
mechanistic target of rapamycin kinase in Human [GtoPdb: 2109] [UniProtKB: P42345]
GtoPdb In an in vitro enzymatic assay. - 5.25 pIC50 5560 nM IC50 ACS Chem Biol (2016) 11: 1537-43 [PMID:27082499]
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta in Human [GtoPdb: 2155] [UniProtKB: O00329]
GtoPdb In an in vitro enzymatic assay. - 6.07 pIC50 856 nM IC50 ACS Chem Biol (2016) 11: 1537-43 [PMID:27082499]
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma in Human [GtoPdb: 2156] [UniProtKB: P48736]
GtoPdb In an in vitro enzymatic assay. - 6.06 pIC50 867 nM IC50 ACS Chem Biol (2016) 11: 1537-43 [PMID:27082499]
serine/threonine kinase 16 in Human [GtoPdb: 2213] [UniProtKB: O75716]
GtoPdb In an in vitro enzymatic inhibition assay. - 6.53 pIC50 295 nM IC50 ACS Chem Biol (2016) 11: 1537-43 [PMID:27082499]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.