catequentinib [Ligand Id: 9601] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| fibroblast growth factor receptor 1 in Human [GtoPdb: 1808] [UniProtKB: P11362] | ||||||||
| GtoPdb | in vitro activity | - | 7.7 | pIC50 | 20 | nM | IC50 | WO2008112407 A1. Spiro substituted compounds as angiogenesis inhibitors (2008) |
| fms related receptor tyrosine kinase 1 in Human [GtoPdb: 1812] [UniProtKB: P17948] | ||||||||
| GtoPdb | In vitro activity | - | 8.4 | pIC50 | 4 | nM | IC50 | WO2008112407 A1. Spiro substituted compounds as angiogenesis inhibitors (2008) |
| kinase insert domain receptor in Human [GtoPdb: 1813] [UniProtKB: P35968] | ||||||||
| GtoPdb | In vitro activity | - | 7.35 | pIC50 | 45 | nM | IC50 | WO2008112407 A1. Spiro substituted compounds as angiogenesis inhibitors (2008) |
| fms related receptor tyrosine kinase 4 in Human [GtoPdb: 1814] [UniProtKB: P35916] | ||||||||
| GtoPdb | In vitro activity | - | 9 | pIC50 | 1 | nM | IC50 | WO2008112407 A1. Spiro substituted compounds as angiogenesis inhibitors (2008) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
