RgIA4 [Ligand Id: 9472] activity data from GtoPdb

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  • nicotinic acetylcholine receptor α9 subunit in Human [GtoPdb: 469] [UniProtKB: Q9UGM1]
  • nicotinic acetylcholine receptor α9 subunit in Rat [GtoPdb: 469] [UniProtKB: P43144]
Created with Highcharts 10.3.3ValuesChart context menunicotinic acetylcholine receptor α9 subunitpKd HumanpKi HumanpIC50 HumanpEC50 HumanpKd RatpKi RatpIC50 RatpEC50 Rat0246810Highcharts.com
  • nicotinic acetylcholine receptor α10 subunit in Human [GtoPdb: 470] [UniProtKB: Q9GZZ6]
  • nicotinic acetylcholine receptor α10 subunit in Rat [GtoPdb: 470] [UniProtKB: Q9JLB5]
Created with Highcharts 10.3.3ValuesChart context menunicotinic acetylcholine receptor α10 subunitpKd HumanpKi HumanpIC50 HumanpEC50 HumanpKd RatpKi RatpIC50 RatpEC50 Rat0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
nicotinic acetylcholine receptor α9 subunit in Human [GtoPdb: 469] [UniProtKB: Q9UGM1]
GtoPdb - - 8.82 pIC50 1.5 nM IC50 Proc Natl Acad Sci USA (2017) 114: E1825-E1832 [PMID:28223528]
nicotinic acetylcholine receptor α9 subunit in Rat [GtoPdb: 469] [UniProtKB: P43144]
GtoPdb - - 9.05 pIC50 0.9 nM IC50 Proc Natl Acad Sci USA (2017) 114: E1825-E1832 [PMID:28223528]
nicotinic acetylcholine receptor α10 subunit in Human [GtoPdb: 470] [UniProtKB: Q9GZZ6]
GtoPdb - - 8.82 pIC50 1.5 nM IC50 Proc Natl Acad Sci USA (2017) 114: E1825-E1832 [PMID:28223528]
nicotinic acetylcholine receptor α10 subunit in Rat [GtoPdb: 470] [UniProtKB: Q9JLB5]
GtoPdb - - 9.05 pIC50 0.9 nM IC50 Proc Natl Acad Sci USA (2017) 114: E1825-E1832 [PMID:28223528]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.