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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| fibroblast growth factor receptor 1 in Human [GtoPdb: 1808] [UniProtKB: P11362] | ||||||||
| GtoPdb | - | - | 8.94 | pIC50 | 1.14 | nM | IC50 | WO2011135376 A1. Pyrazolyl quinazoline kinase inhibitors. (2011) |
| fibroblast growth factor receptor 2 in Human [GtoPdb: 1809] [UniProtKB: P21802] | ||||||||
| GtoPdb | - | - | 8.64 | pIC50 | 2.29 | nM | IC50 | WO2011135376 A1. Pyrazolyl quinazoline kinase inhibitors. (2011) |
| fibroblast growth factor receptor 3 in Human [GtoPdb: 1810] [UniProtKB: P22607] | ||||||||
| GtoPdb | - | - | 8.52 | pIC50 | 3.02 | nM | IC50 | WO2011135376 A1. Pyrazolyl quinazoline kinase inhibitors. (2011) |
| fibroblast growth factor receptor 4 in Human [GtoPdb: 1811] [UniProtKB: P22455] | ||||||||
| GtoPdb | - | - | 8.25 | pIC50 | 5.62 | nM | IC50 | WO2011135376 A1. Pyrazolyl quinazoline kinase inhibitors. (2011) |
| kinase insert domain receptor in Human [GtoPdb: 1813] [UniProtKB: P35968] | ||||||||
| GtoPdb | - | - | 7.44 | pIC50 | 36.3 | nM | IC50 | WO2011135376 A1. Pyrazolyl quinazoline kinase inhibitors. (2011) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.