(S)-ARN2508 [Ligand Id: 8999] activity data from GtoPdb

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  • COX-1 in Human [GtoPdb: 1375] [UniProtKB: P23219]
  • This target only has 0 pki data point
1 _lig_chart_1 COX-1 Human
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  • COX-2 in Human [GtoPdb: 1376] [UniProtKB: P35354]
  • This target only has 0 pki data point
2 _lig_chart_2 COX-2 Human
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  • Fatty acid amide hydrolase in Human [GtoPdb: 1400] [UniProtKB: O00519]
  • This target only has 0 pki data point
3 _lig_chart_3 Fatty acid amide hydrolase Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
COX-1 in Human [GtoPdb: 1375] [UniProtKB: P23219]
GtoPdb - - 9.54 pIC50 0.29 nM IC50 Eur J Med Chem (2016) 109: 216-37 [PMID:26774927]
COX-2 in Human [GtoPdb: 1376] [UniProtKB: P35354]
GtoPdb - - 7.92 pIC50 12 nM IC50 Eur J Med Chem (2016) 109: 216-37 [PMID:26774927]
Fatty acid amide hydrolase in Human [GtoPdb: 1400] [UniProtKB: O00519]
GtoPdb - - 8.03 pIC50 9.4 nM IC50 Eur J Med Chem (2016) 109: 216-37 [PMID:26774927]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.