samotolisib [Ligand Id: 8918] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| mechanistic target of rapamycin kinase in Human [GtoPdb: 2109] [UniProtKB: P42345] | ||||||||
| GtoPdb | - | - | 6.78 | pIC50 | 165 | nM | IC50 | US8440829 B2. PI3 kinase/mTOR dual inhibitor. (2013) |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha in Human [GtoPdb: 2153] [UniProtKB: P42336] | ||||||||
| GtoPdb | - | - | 8.21 | pIC50 | 6.1 | nM | IC50 | US8440829 B2. PI3 kinase/mTOR dual inhibitor. (2013) |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit beta in Human [GtoPdb: 2154] [UniProtKB: P42338] | ||||||||
| GtoPdb | - | - | 7.11 | pIC50 | 78 | nM | IC50 | US8440829 B2. PI3 kinase/mTOR dual inhibitor. (2013) |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta in Human [GtoPdb: 2155] [UniProtKB: O00329] | ||||||||
| GtoPdb | - | - | 7.42 | pIC50 | 38 | nM | IC50 | US8440829 B2. PI3 kinase/mTOR dual inhibitor. (2013) |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma in Human [GtoPdb: 2156] [UniProtKB: P48736] | ||||||||
| GtoPdb | - | - | 7.62 | pIC50 | 23.8 | nM | IC50 | US8440829 B2. PI3 kinase/mTOR dual inhibitor. (2013) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
