GLPG0974 [Ligand Id: 8417] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| FFA2 receptor in Human [GtoPdb: 226] [UniProtKB: O15552] | ||||||||
| GtoPdb | Inhibition of sodium acetate-induced calcium flux via the FFA2 receptor. | - | 8.05 | pIC50 | 9 | nM | IC50 |
J Med Chem (2014) 57: 10044-57 [PMID:25380412]; Br J Clin Pharmacol (2016) 82: 139-48 [PMID:26852904] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
