PI-3065 [Ligand Id: 8242] activity data from GtoPdb

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  • phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit beta in Human [GtoPdb: 2154] [UniProtKB: P42338]
Created with Highcharts 10.3.3ValuesChart context menuphosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit betapKd HumanpKi HumanpIC50 HumanpEC50 Human01234567Highcharts.com
  • phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta in Human [GtoPdb: 2155] [UniProtKB: O00329]
Created with Highcharts 10.3.3ValuesChart context menuphosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit deltapKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit beta in Human [GtoPdb: 2154] [UniProtKB: P42338]
GtoPdb - - 5.97 pIC50 1078 nM IC50 Nature (2014) 510: 407-11 [PMID:24919154]
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta in Human [GtoPdb: 2155] [UniProtKB: O00329]
GtoPdb - - 7.82 pIC50 15 nM IC50 Nature (2014) 510: 407-11 [PMID:24919154]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.