I-CBP112 [Ligand Id: 8236] activity data from GtoPdb

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  • CREB binding lysine acetyltransferase in Human [GtoPdb: 2734] [UniProtKB: Q92793]
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  • EP300 lysine acetyltransferase in Human [GtoPdb: 2735] [UniProtKB: Q09472]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
CREB binding lysine acetyltransferase in Human [GtoPdb: 2734] [UniProtKB: Q92793]
GtoPdb Isothermal titration calorimetry (ITC) assay. - 6.85 pKd 142 nM Kd I-CBP112 A CREBBP/EP300-selective chemical probe. thesgc.org
EP300 lysine acetyltransferase in Human [GtoPdb: 2735] [UniProtKB: Q09472]
GtoPdb Isothermal titration calorimetry (ITC) assay. - 6.2 pKd 625 nM Kd I-CBP112 A CREBBP/EP300-selective chemical probe. thesgc.org

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.