α-CGRP-(8-37) (human) [Ligand Id: 700] activity data from GtoPdb

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  • AMY1 receptor in Human [GtoPdb: 44]
Created with Highcharts 10.3.3ValuesChart context menuAMY1 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human0Highcharts.com
  • AMY3 receptor in Human [GtoPdb: 46]
Created with Highcharts 10.3.3ValuesChart context menuAMY3 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human0Highcharts.com
  • CGRP receptor in Human [GtoPdb: 48]
Created with Highcharts 10.3.3ValuesChart context menuCGRP receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human024681012Highcharts.com
  • AM1 receptor in Human [GtoPdb: 49]
Created with Highcharts 10.3.3ValuesChart context menuAM1 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
  • AM2 receptor in Human [GtoPdb: 50]
Created with Highcharts 10.3.3ValuesChart context menuAM2 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
AMY1 receptor in Human [GtoPdb: 44]
AMY3 receptor in Human [GtoPdb: 46]
CGRP receptor in Human [GtoPdb: 48]
GtoPdb - - 9.6 pKi - - - Nature (1998) 393: 333-9 [PMID:9620797];
Mol Cell Biochem (2001) 224: 123-33 [PMID:11693189]
AM1 receptor in Human [GtoPdb: 49]
GtoPdb - - 7 pKi - - - Nature (1998) 393: 333-9 [PMID:9620797];
Mol Cell Biochem (2001) 224: 123-33 [PMID:11693189]
AM2 receptor in Human [GtoPdb: 50]
GtoPdb - - 6.5 pKi - - - Mol Cell Biochem (2001) 224: 123-33 [PMID:11693189];
Mol Pharmacol (1999) 55: 1054-1059 [PMID:10347248]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.