VPC03090-P [Ligand Id: 6992] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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| S1P1 receptor in Human [GtoPdb: 275] [UniProtKB: P21453] | ||||||||
| GtoPdb | - | - | 7.68 | pKi | 21 | nM | Ki | J Pharmacol Exp Ther (2011) 338: 879-89 [PMID:21632869] |
| S1P1 receptor in Mouse [GtoPdb: 275] [UniProtKB: O08530] | ||||||||
| GtoPdb | - | - | 7.85 | pKi | 14 | nM | Ki | J Pharmacol Exp Ther (2011) 338: 879-89 [PMID:21632869] |
| S1P3 receptor in Human [GtoPdb: 277] [UniProtKB: Q99500] | ||||||||
| GtoPdb | - | - | 7.29 | pKi | 51 | nM | Ki | J Pharmacol Exp Ther (2011) 338: 879-89 [PMID:21632869] |
| S1P4 receptor in Human [GtoPdb: 278] [UniProtKB: O95977] | ||||||||
| GtoPdb | - | - | 7.76 | pKd | 17.3 | nM | Kd | J Pharmacol Exp Ther (2011) 338: 879-89 [PMID:21632869] |
| GtoPdb | - | - | 7.75 | pEC50 | 17.7 | nM | EC50 | J Pharmacol Exp Ther (2011) 338: 879-89 [PMID:21632869] |
| S1P5 receptor in Human [GtoPdb: 279] [UniProtKB: Q9H228] | ||||||||
| GtoPdb | - | - | 8.64 | pKd | 2.3 | nM | Kd | J Pharmacol Exp Ther (2011) 338: 879-89 [PMID:21632869] |
| GtoPdb | - | - | 8.62 | pEC50 | 2.4 | nM | EC50 | J Pharmacol Exp Ther (2011) 338: 879-89 [PMID:21632869] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
