YSFKPMPLaR [Ligand Id: 5776] activity data from GtoPdb

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  • C3a receptor in Human [GtoPdb: 31] [UniProtKB: Q16581]
Created with Highcharts 10.3.3ValuesChart context menuC3a receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
  • C5a1 receptor in Human [GtoPdb: 32] [UniProtKB: P21730]
Created with Highcharts 10.3.3ValuesChart context menuC5a1 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
C3a receptor in Human [GtoPdb: 31] [UniProtKB: Q16581]
GtoPdb - - 6.7 pEC50 220 nM EC50 J Med Chem (2010) 53: 4938-48 [PMID:20527893]
C5a1 receptor in Human [GtoPdb: 32] [UniProtKB: P21730]
GtoPdb - - 6.7 pIC50 200 nM IC50 J Med Chem (1997) 40: 877-84 [PMID:9083476]
GtoPdb - - 5.5 pEC50 3240 nM EC50 Inflammation (2001) 25: 171-7 [PMID:11403208]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.