[3H]MK-912 [Ligand Id: 527] activity data from GtoPdb
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| α2A-adrenoceptor in Human [GtoPdb: 25] [UniProtKB: P08913] | ||||||||
| GtoPdb | - | - | 8.9 | pKd | 1.25 | nM | Kd | J Pharmacol Exp Ther (1994) 271: 1558-65 [PMID:7996470] |
| α2B-adrenoceptor in Human [GtoPdb: 26] [UniProtKB: P18089] | ||||||||
| GtoPdb | - | - | 8.9 | pKd | 1.36 | nM | Kd | J Pharmacol Exp Ther (1994) 271: 1558-65 [PMID:7996470] |
| α2C-adrenoceptor in Human [GtoPdb: 27] [UniProtKB: P18825] | ||||||||
| GtoPdb | - | - | 10.1 | pKd | 0.09 | nM | Kd | J Pharmacol Exp Ther (1994) 271: 1558-65 [PMID:7996470] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
