Cu2+ [Ligand Id: 4164] activity data from GtoPdb
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| glycine receptor α1 subunit in Human [GtoPdb: 423] [UniProtKB: P23415] | ||||||||
| GtoPdb | - | - | 5.4 | pIC50 | 4000 | nM | IC50 | |
| glycine receptor α2 subunit in Human [GtoPdb: 424] [UniProtKB: P23416] | ||||||||
| GtoPdb | - | - | 4.8 | pIC50 | 17000 | nM | IC50 | |
| glycine receptor α3 subunit in Human [GtoPdb: 425] [UniProtKB: O75311] | ||||||||
| GtoPdb | - | - | 5 | pIC50 | 9000 | nM | IC50 | |
| TRPA1 in Human [GtoPdb: 485] [UniProtKB: O75762] | ||||||||
| GtoPdb | Sodium imaging | - | 5.89 | pEC50 | 1300 | nM | EC50 |
Proc Natl Acad Sci USA (2009) 106: 8374-9 [PMID:19416844]; Mol Pain (2013) 9: 7 [PMID:23448290] |
| TRPA1 in Mouse [GtoPdb: 485] [UniProtKB: Q8BLA8] | ||||||||
| GtoPdb | - | - | 6.22 | pEC50 | 600 | nM | EC50 |
Proc Natl Acad Sci USA (2009) 106: 8374-9 [PMID:19416844]; Mol Pain (2013) 9: 7 [PMID:23448290] |
| ZAC in Human [GtoPdb: 587] [UniProtKB: Q401N2] | ||||||||
| GtoPdb | - | - | 5.4 | pEC50 | - | - | - | Biochem Pharmacol (2016) 103: 109-17 [PMID:26872532] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
