Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
---|---|---|---|---|---|---|---|---|
M1 receptor in Human [GtoPdb: 13] [UniProtKB: P11229] | ||||||||
GtoPdb | - | - | 7.7 | pKi | - | - | - | Biochem Pharmacol (1996) 52: 643-58 [PMID:8759038] |
M1 receptor in Rat [GtoPdb: 13] [UniProtKB: P08482] | ||||||||
GtoPdb | - | - | 7.9 | pKi | - | - | - |
Life Sci (1992) 51: 955-71 [PMID:1325587]; Mol Pharmacol (1989) 35: 469-76 [PMID:2704370] |
M2 receptor in Human [GtoPdb: 14] [UniProtKB: P08172] | ||||||||
GtoPdb | - | - | 6.8 | pKi | - | - | - |
Biochem Pharmacol (1996) 52: 643-58 [PMID:8759038]; Mol Pharmacol (1989) 35: 469-76 [PMID:2704370]; J Pharmacol Exp Ther (1998) 284: 500-7 [PMID:9454790] |
M2 receptor in Rat [GtoPdb: 14] [UniProtKB: P10980] | ||||||||
GtoPdb | - | - | 6.8 | pKi | - | - | - |
Life Sci (1992) 51: 955-71 [PMID:1325587]; J Pharmacol Exp Ther (1998) 284: 500-7 [PMID:9454790] |
M3 receptor in Human [GtoPdb: 15] [UniProtKB: P20309] | ||||||||
GtoPdb | - | - | 8 | pKi | - | - | - |
Biochem Pharmacol (1996) 52: 643-58 [PMID:8759038]; Mol Pharmacol (1989) 35: 469-76 [PMID:2704370] |
M4 receptor in Human [GtoPdb: 16] [UniProtKB: P08173] | ||||||||
GtoPdb | - | - | 7.7 | pKi | - | - | - |
Biochem Pharmacol (1996) 52: 643-58 [PMID:8759038]; Mol Pharmacol (1989) 35: 469-76 [PMID:2704370] |
M4 receptor in Rat [GtoPdb: 16] [UniProtKB: P08485] | ||||||||
GtoPdb | - | - | 7.7 | pKi | - | - | - | Life Sci (1992) 51: 955-71 [PMID:1325587] |
M5 receptor in Human [GtoPdb: 17] [UniProtKB: P08912] | ||||||||
GtoPdb | - | - | 7.2 | pKi | - | - | - |
Biochem Pharmacol (1996) 52: 643-58 [PMID:8759038]; Mol Pharmacol (1989) 35: 469-76 [PMID:2704370] |
M5 receptor in Rat [GtoPdb: 17] [UniProtKB: P08911] | ||||||||
GtoPdb | - | - | 7.4 | pKi | - | - | - | Life Sci (1992) 51: 955-71 [PMID:1325587] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.