WJH-C19 [Ligand Id: 14350] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha in Human [GtoPdb: 2153] [UniProtKB: P42336]
There should be some charts here, you may need to enable JavaScript!
  • receptor interacting serine/threonine kinase 1 in Human [GtoPdb: 2189] [UniProtKB: Q13546]
There should be some charts here, you may need to enable JavaScript!
  • receptor interacting serine/threonine kinase 2 in Human [GtoPdb: 2190] [UniProtKB: O43353]
There should be some charts here, you may need to enable JavaScript!
  • receptor interacting serine/threonine kinase 3 in Human [GtoPdb: 2191] [UniProtKB: Q9Y572]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha in Human [GtoPdb: 2153] [UniProtKB: P42336]
GtoPdb - - 5 pIC50 10000 nM IC50 J Med Chem (2026) 69: 3252-3288 [PMID:41628914]
receptor interacting serine/threonine kinase 1 in Human [GtoPdb: 2189] [UniProtKB: Q13546]
GtoPdb - - 8.24 pIC50 5.7 nM IC50 J Med Chem (2026) 69: 3252-3288 [PMID:41628914]
receptor interacting serine/threonine kinase 2 in Human [GtoPdb: 2190] [UniProtKB: O43353]
GtoPdb - - 6 pIC50 >1000 nM IC50 J Med Chem (2026) 69: 3252-3288 [PMID:41628914]
receptor interacting serine/threonine kinase 3 in Human [GtoPdb: 2191] [UniProtKB: Q9Y572]
GtoPdb - - 6 pIC50 >1000 nM IC50 J Med Chem (2026) 69: 3252-3288 [PMID:41628914]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.