SK5527 [Ligand Id: 14285] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| aurora kinase A in Human [GtoPdb: 1936] [UniProtKB: O14965] | ||||||||
| GtoPdb | - | - | 8.7 | pKi | 2 | nM | Ki | J Med Chem (2025) : [PMID:41252673] |
| GtoPdb | Determined as displacement of tracer from NanoLuc-AURKA in a NanoBRET assay | - | 7.7 | pIC50 | 20 | nM | IC50 | J Med Chem (2025) : [PMID:41252673] |
| cereblon in Human [GtoPdb: 3086] [UniProtKB: Q96SW2] | ||||||||
| GtoPdb | - | - | 5.95 | pKi | 1133 | nM | Ki | J Med Chem (2025) : [PMID:41252673] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
