compound 35 [PMID: 41114343] [Ligand Id: 14248] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| apelin receptor in Human [GtoPdb: 36] [UniProtKB: P35414] | ||||||||
| GtoPdb | Agonist potency determined in a β-arrestin2 recruitment assay | - | 6.52 | pEC50 | 301 | nM | EC50 | J Med Chem (2025) 68: 22312-22332 [PMID:41114538] |
| GtoPdb | Agonist potency determined in a cAMP accumulation assay | - | 8 | pEC50 | 10 | nM | EC50 | J Med Chem (2025) 68: 22312-22332 [PMID:41114538] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
