ontunisertib [Ligand Id: 13846] activity data from GtoPdb
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| transforming growth factor beta receptor 1 in Human [GtoPdb: 1788] [UniProtKB: P36897] | ||||||||
| GtoPdb | Determined in a biochemical ADP-Glo kinase inhibition assay | - | 7 | pIC50 | <100 | nM | IC50 | WO2021105317A1. Benzylamide derivatives as inhibitors of transforming growth factor-beta receptor i/alk5 (2021) |
| GtoPdb | Determined in a cellular assay using TGF-stimulated A549 cells | - | 7 | pIC50 | 100 | nM | IC50 | WO2021105317A1. Benzylamide derivatives as inhibitors of transforming growth factor-beta receptor i/alk5 (2021) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
