tosposertib [Ligand Id: 13752] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • transforming growth factor beta receptor 1 in Human [GtoPdb: 1788] [UniProtKB: P36897]
Created with Highcharts 10.3.3ValuesChart context menutransforming growth factor beta receptor 1pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
transforming growth factor beta receptor 1 in Human [GtoPdb: 1788] [UniProtKB: P36897]
GtoPdb - - 7.94 pIC50 11.5 nM IC50 US10155763B2. 2-pyridyl substituted imidazoles as ALK5 and/or ALK4 inhibitors (2018)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.