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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| MC1 receptor in Human [GtoPdb: 282] [UniProtKB: Q01726] | ||||||||
| GtoPdb | - | - | 8.4 | pIC50 | - | - | - | Eur J Pharmacol (2002) 440: 141-57 [PMID:12007532] |
| MC3 receptor in Human [GtoPdb: 284] [UniProtKB: P41968] | ||||||||
| GtoPdb | - | - | 8.4 | pKi | - | - | - |
J Biol Chem (1999) 274: 16853-60 [PMID:10358030]; Eur J Pharmacol (1999) 378: 249-258 [PMID:10493100] |
| MC4 receptor in Human [GtoPdb: 285] [UniProtKB: P32245] | ||||||||
| GtoPdb | - | - | 8 | pKi | - | - | - |
Eur J Pharmacol (1999) 378: 249-258 [PMID:10493100]; Biochemistry (2000) 39: 14900-11 [PMID:11101306] |
| MC5 receptor in Human [GtoPdb: 286] [UniProtKB: P33032] | ||||||||
| GtoPdb | - | - | 6.9 | pKd | - | - | - | Eur J Pharmacol (2002) 440: 141-57 [PMID:12007532] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.