 
 
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
| 
 There should be some charts here, you may need to enable JavaScript! | 
| There should be some charts here, you may need to enable JavaScript! | 
| There should be some charts here, you may need to enable JavaScript! | 
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference | 
|---|---|---|---|---|---|---|---|---|
| enhancer of zeste 2 polycomb repressive complex 2 subunit in Human [GtoPdb: 2654] [UniProtKB: Q15910] | ||||||||
| GtoPdb | - | - | 6.6 | pIC50 | 250 | nM | IC50 | J Med Chem (2023) 66: 1634-1651 [PMID:36642961] | 
| nuclear receptor binding SET domain protein 1 in Human [GtoPdb: 2696] [UniProtKB: Q96L73] | ||||||||
| GtoPdb | - | - | 6.16 | pIC50 | 690 | nM | IC50 | J Med Chem (2023) 66: 1634-1651 [PMID:36642961] | 
| nuclear receptor binding SET domain protein 2 in Human [GtoPdb: 3220] [UniProtKB: O96028] | ||||||||
| GtoPdb | - | - | 6.64 | pIC50 | 230 | nM | IC50 | J Med Chem (2023) 66: 1634-1651 [PMID:36642961] | 
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.