TAK-020 [Ligand Id: 11730] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Bruton tyrosine kinase in Human [GtoPdb: 1948] [UniProtKB: Q06187] | ||||||||
| GtoPdb | - | - | 8.7 | pIC50 | <1.99 | nM | IC50 | J Med Chem (2021) 64: 12893-12902 [PMID:34448571] |
| LCK proto-oncogene, Src family tyrosine kinase in Human [GtoPdb: 2053] [UniProtKB: P06239] | ||||||||
| GtoPdb | - | - | 6 | pIC50 | 1000 | nM | IC50 | J Med Chem (2021) 64: 12893-12902 [PMID:34448571] |
| SRC proto-oncogene, non-receptor tyrosine kinase in Human [GtoPdb: 2206] [UniProtKB: P12931] | ||||||||
| GtoPdb | - | - | 6.2 | pIC50 | 631 | nM | IC50 | J Med Chem (2021) 64: 12893-12902 [PMID:34448571] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
