nemtabrutinib [Ligand Id: 11413] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| BLK proto-oncogene, Src family tyrosine kinase in Human [GtoPdb: 1940] [UniProtKB: P51451] | ||||||||
| GtoPdb | - | - | 8.01 | pIC50 | 9.7 | nM | IC50 | Cancer Discov (2018) 8: 1300-1315 [PMID:30093506] |
| BMX non-receptor tyrosine kinase in Human [GtoPdb: 1942] [UniProtKB: P51813] | ||||||||
| GtoPdb | - | - | 8.28 | pIC50 | 5.2 | nM | IC50 | Cancer Discov (2018) 8: 1300-1315 [PMID:30093506] |
| Bruton tyrosine kinase in Human [GtoPdb: 1948] [UniProtKB: Q06187] | ||||||||
| GtoPdb | Inhibition of enzyme activity in a biochemical assay | - | 8.6 | pIC50 | 2.5 | nM | IC50 | Cancer Discov (2018) 8: 1300-1315 [PMID:30093506] |
| tec protein tyrosine kinase in Human [GtoPdb: 2238] [UniProtKB: P42680] | ||||||||
| GtoPdb | - | - | 8.24 | pIC50 | 5.8 | nM | IC50 | Cancer Discov (2018) 8: 1300-1315 [PMID:30093506] |
| YES proto-oncogene 1, Src family tyrosine kinase in Human [GtoPdb: 2284] [UniProtKB: P07947] | ||||||||
| GtoPdb | - | - | 8.38 | pIC50 | 4.2 | nM | IC50 | Cancer Discov (2018) 8: 1300-1315 [PMID:30093506] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
