compound 71 [WO2018191577A1] [Ligand Id: 11203] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • Bruton tyrosine kinase in Human [GtoPdb: 1948] [UniProtKB: Q06187]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Bruton tyrosine kinase in Human [GtoPdb: 1948] [UniProtKB: Q06187]
GtoPdb Measuring inhibition of substrate peptide phosphorylation in the presence of active BTK enzyme, ATP, and inhibitor. - 9 pIC50 <1 nM IC50 WO2018191577A1. Benzoazepine analogs as inhibiting agents for bruton's tyrosine kinase (2018)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.