dalpiciclib [Ligand Id: 11189] activity data from GtoPdb

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  • cyclin dependent kinase 4 in Human [GtoPdb: 1976] [UniProtKB: P11802]
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  • cyclin dependent kinase 6 in Human [GtoPdb: 1978] [UniProtKB: Q00534]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
cyclin dependent kinase 4 in Human [GtoPdb: 1976] [UniProtKB: P11802]
GtoPdb - - 7.96 pIC50 11 nM IC50 WO2014183520A1. Thiophene miazines derivate, preparation method therefor, and medical application thereof (2014)
cyclin dependent kinase 6 in Human [GtoPdb: 1978] [UniProtKB: Q00534]
GtoPdb - - 8.22 pIC50 6 nM IC50 WO2014183520A1. Thiophene miazines derivate, preparation method therefor, and medical application thereof (2014)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.