BSJ-03-204 [Ligand Id: 10530] activity data from GtoPdb

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  • cyclin dependent kinase 4 in Human [GtoPdb: 1976] [UniProtKB: P11802]
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  • cyclin dependent kinase 6 in Human [GtoPdb: 1978] [UniProtKB: Q00534]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
cyclin dependent kinase 4 in Human [GtoPdb: 1976] [UniProtKB: P11802]
GtoPdb Inhibition of CDK4/cyclin D1 kinase activity in a biochemical assay. - 7.57 pIC50 26.9 nM IC50 Angew Chem Int Ed Engl (2019) 58: 6321-6326 [PMID:30802347]
cyclin dependent kinase 6 in Human [GtoPdb: 1978] [UniProtKB: Q00534]
GtoPdb Inhibition of CDK6/cyclin D1 kinase activity in a biochemical assay. - 7.98 pIC50 10.4 nM IC50 Angew Chem Int Ed Engl (2019) 58: 6321-6326 [PMID:30802347]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.