BSJ-03-204 [Ligand Id: 10530] activity data from GtoPdb

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  • cyclin dependent kinase 4 in Human [GtoPdb: 1976] [UniProtKB: P11802]
Created with Highcharts 10.3.3ValuesChart context menucyclin dependent kinase 4pKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
  • cyclin dependent kinase 6 in Human [GtoPdb: 1978] [UniProtKB: Q00534]
Created with Highcharts 10.3.3ValuesChart context menucyclin dependent kinase 6pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
cyclin dependent kinase 4 in Human [GtoPdb: 1976] [UniProtKB: P11802]
GtoPdb Inhibition of CDK4/cyclin D1 kinase activity in a biochemical assay. - 7.57 pIC50 26.9 nM IC50 Angew Chem Int Ed Engl (2019) 58: 6321-6326 [PMID:30802347]
cyclin dependent kinase 6 in Human [GtoPdb: 1978] [UniProtKB: Q00534]
GtoPdb Inhibition of CDK6/cyclin D1 kinase activity in a biochemical assay. - 7.98 pIC50 10.4 nM IC50 Angew Chem Int Ed Engl (2019) 58: 6321-6326 [PMID:30802347]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.