neolymphostin A [Ligand Id: 10151] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| LCK proto-oncogene, Src family tyrosine kinase in Human [GtoPdb: 2053] [UniProtKB: P06239] | ||||||||
| GtoPdb | - | - | 5.34 | pKd | 4600 | nM | Kd | J Med Chem (2018) 61: 10463-10472 [PMID:30380865] |
| mechanistic target of rapamycin kinase in Human [GtoPdb: 2109] [UniProtKB: P42345] | ||||||||
| GtoPdb | Determined using an active-site dependent competition binding assay. | - | 8 | pKd | 10 | nM | Kd | J Med Chem (2018) 61: 10463-10472 [PMID:30380865] |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha in Human [GtoPdb: 2153] [UniProtKB: P42336] | ||||||||
| GtoPdb | Determined using an active-site dependent competition binding assay. | - | 9.06 | pKd | 0.88 | nM | Kd | J Med Chem (2018) 61: 10463-10472 [PMID:30380865] |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit beta in Human [GtoPdb: 2154] [UniProtKB: P42338] | ||||||||
| GtoPdb | Determined using an active-site dependent competition binding assay. | - | 8.24 | pKd | 5.7 | nM | Kd | J Med Chem (2018) 61: 10463-10472 [PMID:30380865] |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta in Human [GtoPdb: 2155] [UniProtKB: O00329] | ||||||||
| GtoPdb | Determined using an active-site dependent competition binding assay. | - | 8.31 | pKd | 4.9 | nM | Kd | J Med Chem (2018) 61: 10463-10472 [PMID:30380865] |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma in Human [GtoPdb: 2156] [UniProtKB: P48736] | ||||||||
| GtoPdb | Determined using an active-site dependent competition binding assay. | - | 8.46 | pKd | 3.5 | nM | Kd | J Med Chem (2018) 61: 10463-10472 [PMID:30380865] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
