BTK inhibitor 16 [PMID: 30122225] [Ligand Id: 10076] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Bruton tyrosine kinase in Human [GtoPdb: 1948] [UniProtKB: Q06187] | ||||||||
| GtoPdb | Using a microfluidic, off-chip mobility shift kinase assay with FITC-AHA-EEPLYWSFPAKKK-NH2 as peptide substrate. | - | 9.15 | pIC50 | 0.7 | nM | IC50 | Bioorg Med Chem Lett (2018) 28: 2939-2944 [PMID:30122225] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
