dual BRD4/PLK1 inhibitor 23 [Ligand Id: 10072] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| bromodomain containing 4 in Human [GtoPdb: 1945] [UniProtKB: O60885] | ||||||||
| GtoPdb | Biochemical inhibition of BRD4-BD1. | - | 7.55 | pIC50 | 28 | nM | IC50 | J Med Chem (2018) 61: 7785-7795 [PMID:30125504] |
| polo like kinase 1 in Human [GtoPdb: 2168] [UniProtKB: P53350] | ||||||||
| GtoPdb | Biochemical inhibition of PLK1. | - | 7.4 | pIC50 | 40 | nM | IC50 | J Med Chem (2018) 61: 7785-7795 [PMID:30125504] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
