Des-AA5-[D-Trp8]SRIF   Click here for help

GtoPdb Ligand ID: 2012

Compound class: Peptide
Comment: Synthetic analogue of somatostatin-14
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
SST1 receptor Hs Agonist Full agonist 8.9 – 9.1 pIC50 - 1
pIC50 8.9 – 9.1 [1]
SST4 receptor Hs Agonist Full agonist 8.7 – 8.9 pIC50 - 1
pIC50 8.7 – 8.9 [1]
SST3 receptor Hs Agonist Full agonist 8.4 – 8.5 pIC50 - 1
pIC50 8.4 – 8.5 [1]
SST5 receptor Hs Agonist Full agonist 8.2 – 8.4 pIC50 - 1
pIC50 8.2 – 8.4 [1]