Des-AA5-[D-Trp8]SRIF [Ligand Id: 2012] activity data from GtoPdb

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  • SST1 receptor in Human [GtoPdb: 355] [UniProtKB: P30872]
Created with Highcharts 10.3.3ValuesChart context menuSST1 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • SST3 receptor in Human [GtoPdb: 357] [UniProtKB: P32745]
Created with Highcharts 10.3.3ValuesChart context menuSST3 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • SST4 receptor in Human [GtoPdb: 358] [UniProtKB: P31391]
Created with Highcharts 10.3.3ValuesChart context menuSST4 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • SST5 receptor in Human [GtoPdb: 359] [UniProtKB: P35346]
Created with Highcharts 10.3.3ValuesChart context menuSST5 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
SST1 receptor in Human [GtoPdb: 355] [UniProtKB: P30872]
GtoPdb - - 9.1 pIC50 - - - J Med Chem (2005) 48: 507-514 [PMID:15658864]
SST3 receptor in Human [GtoPdb: 357] [UniProtKB: P32745]
GtoPdb - - 8.5 pIC50 - - - J Med Chem (2005) 48: 507-514 [PMID:15658864]
SST4 receptor in Human [GtoPdb: 358] [UniProtKB: P31391]
GtoPdb - - 8.9 pIC50 - - - J Med Chem (2005) 48: 507-514 [PMID:15658864]
SST5 receptor in Human [GtoPdb: 359] [UniProtKB: P35346]
GtoPdb - - 8.4 pIC50 - - - J Med Chem (2005) 48: 507-514 [PMID:15658864]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.