compound 29 [Moslin et al., 2017] [Ligand Id: 9992] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| phosphodiesterase 4D in Human [GtoPdb: 1303] [UniProtKB: Q08499] | ||||||||
| GtoPdb | Binding affinity calculated be measuring displacement of [3H]cAMP binding to purified recombinant His-Tb-hPDE4D2. | - | 7.37 | pIC50 | 43 | nM | IC50 | Medchemcomm (2017) 8: 700-712 [PMID:30108788] |
| tyrosine kinase 2 in Human [GtoPdb: 2269] [UniProtKB: P29597] | ||||||||
| GtoPdb | Measuring binding to the JH2 pseudokinase domain of human TYK2. | - | 8.4 | pIC50 | 4 | nM | IC50 | Medchemcomm (2017) 8: 700-712 [PMID:30108788] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
