PF‐06526290 [Ligand Id: 9980] activity data from GtoPdb

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  • Nav1.3 in Human [GtoPdb: 580] [UniProtKB: Q9NY46]
Created with Highcharts 10.3.3ValuesChart context menuNav1.3pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • Nav1.7 in Human [GtoPdb: 584] [UniProtKB: Q15858]
Created with Highcharts 10.3.3ValuesChart context menuNav1.7pKd HumanpKi HumanpIC50 HumanpEC50 Human024681012Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Nav1.3 in Human [GtoPdb: 580] [UniProtKB: Q9NY46]
GtoPdb - - 8.96 pEC50 1.1 nM EC50 Br J Pharmacol (2018) 175: 2926-2939 [PMID:29791744]
Nav1.7 in Human [GtoPdb: 584] [UniProtKB: Q15858]
GtoPdb - - 9.57 pEC50 0.27 nM EC50 Br J Pharmacol (2018) 175: 2926-2939 [PMID:29791744]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.