SH045 [Ligand Id: 9968] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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| TRPC3 in Human [GtoPdb: 488] [UniProtKB: Q13507] | ||||||||
| GtoPdb | Measuring inhibition of calcium flux in HEK293 cells expressing hTRPC3, in a FLIPR assay. | - | 6.08 | pIC50 | 840 | nM | IC50 | ChemMedChem (2018) 13: 1028-1035 [PMID:29522264] |
| TRPC6 in Human [GtoPdb: 491] [UniProtKB: Q9Y210] | ||||||||
| GtoPdb | Measuring inhibition of calcium flux in HEK293 cells expressing hTRPC6, in a FLIPR assay. | - | 7.2 | pIC50 | 63 | nM | IC50 | ChemMedChem (2018) 13: 1028-1035 [PMID:29522264] |
| TRPC7 in Human [GtoPdb: 492] [UniProtKB: Q9HCX4] | ||||||||
| GtoPdb | Measuring inhibition of calcium flux in HEK293 cells expressing hTRPC7, in a FLIPR assay. | - | 6.66 | pIC50 | 220 | nM | IC50 | ChemMedChem (2018) 13: 1028-1035 [PMID:29522264] |
| GtoPdb | - | - | 7.7 | pIC50 | ~20 | nM | IC50 | ChemMedChem (2018) 13: 1028-1035 [PMID:29522264] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
