AZD9567 [Ligand Id: 9812] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Glucocorticoid receptor in Human [GtoPdb: 625] [UniProtKB: P04150] | ||||||||
| GtoPdb | Binding to human GR in vitro . | - | 8.42 | pIC50 | 3.8 | nM | IC50 | J Med Chem (2018) 61: 1785-1799 [PMID:29424542] |
| GtoPdb | In a cellular transactivation assay. | - | 7.96 | pEC50 | 11 | nM | EC50 | J Med Chem (2018) 61: 1785-1799 [PMID:29424542] |
| Mineralocorticoid receptor in Human [GtoPdb: 626] [UniProtKB: P08235] | ||||||||
| GtoPdb | - | - | 4.42 | pIC50 | >38000 | nM | IC50 | J Med Chem (2018) 61: 1785-1799 [PMID:29424542] |
| Progesterone receptor in Human [GtoPdb: 627] [UniProtKB: P06401] | ||||||||
| GtoPdb | - | - | 5.28 | pIC50 | 5300 | nM | IC50 | J Med Chem (2018) 61: 1785-1799 [PMID:29424542] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
