AZD9567 [Ligand Id: 9812] activity data from GtoPdb

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  • Glucocorticoid receptor in Human [GtoPdb: 625] [UniProtKB: P04150]
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  • Mineralocorticoid receptor in Human [GtoPdb: 626] [UniProtKB: P08235]
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  • Progesterone receptor in Human [GtoPdb: 627] [UniProtKB: P06401]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Glucocorticoid receptor in Human [GtoPdb: 625] [UniProtKB: P04150]
GtoPdb Binding to human GR in vitro . - 8.42 pIC50 3.8 nM IC50 J. Med. Chem. (2018) 61: 1785-1799 [PMID:29424542]
GtoPdb In a cellular transactivation assay. - 7.96 pEC50 11 nM EC50 J. Med. Chem. (2018) 61: 1785-1799 [PMID:29424542]
Mineralocorticoid receptor in Human [GtoPdb: 626] [UniProtKB: P08235]
GtoPdb - - 4.42 pIC50 >38000 nM IC50 J. Med. Chem. (2018) 61: 1785-1799 [PMID:29424542]
Progesterone receptor in Human [GtoPdb: 627] [UniProtKB: P06401]
GtoPdb - - 5.28 pIC50 5300 nM IC50 J. Med. Chem. (2018) 61: 1785-1799 [PMID:29424542]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.